What is the significance of structure-activity relationship (SAR) in drug synthe
Practice Questions
Q1
What is the significance of structure-activity relationship (SAR) in drug synthesis?
It helps in predicting drug interactions
It aids in optimizing drug potency
It determines the drug's market price
It is irrelevant to drug design
Questions & Step-by-Step Solutions
What is the significance of structure-activity relationship (SAR) in drug synthesis?
Step 1: Understand that structure-activity relationship (SAR) is a concept that studies how the chemical structure of a compound affects its biological activity.
Step 2: Recognize that in drug synthesis, SAR helps scientists identify which parts of a molecule are important for its effectiveness as a drug.
Step 3: Learn that by modifying the structure of a drug, researchers can improve its potency, meaning it works better at lower doses.
Step 4: Realize that SAR also helps in increasing the efficacy of a drug, which means it can produce a desired effect more reliably.
Step 5: Conclude that understanding SAR is crucial for developing new drugs that are safer and more effective for patients.
